APX-115
目录号: A18737
Nox 抑制剂
APX-115(Ewha-18278)是一种有效的口服全能 NADPH氧化酶(Nox)抑制剂,其Ki值分别针对Nox1、Nox2和Nox4为1.08 μM、0.57 μM和0.63 μM。APX-115能有效预防肾脏损伤。
Discription | APX-115 (Ewha-18278) is a potent, orally active pan NADPH oxidase (Nox) inhibitor with Ki values of 1.08 μM, 0.57 μM, and 0.63 μM for Nox1, Nox2 and Nox4, respectively. APX-115 effectively prevents kidney injury. |
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目录号 | A18737 |
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分子式 | C17H18ClN3O |
分子量 | 315.8 |
CAS号 | 1395946-75-4 |
SMILES | OC1=C(CCC)C(C2=CC=CC=C2)=NN1C3=NC=CC=C3.Cl |
其他名称 | APX 115, APX115 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2