AS2863619
目录号: A22338
CDK8 and CDK19 抑制剂
AS2863619 是一种强效的、口服活性的环依赖性激酶8(CDK8)和CDK19抑制剂,其半抑制浓度(IC50)分别为0.61纳摩尔和4.28纳摩尔。
Discription | AS2863619 is a potent, orally active cyclin-dependent kinase 8 (CDK8) and CDK19 inhibitor with IC50s of 0.61 nM and 4.28 nM, respectively. |
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目录号 | A22338 |
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分子式 | C16H14Cl2N8O |
分子量 | 405.24 |
CAS号 | 2241300-51-4 |
SMILES | NC1=NON=C1C(N2C3=CC=C4N=C(C)NC4=C3)=NC5=C2C=CN=C5.[H]Cl.[H]Cl |
其他名称 | AS 2863619,AS-2863619 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2