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Asenapine maleate

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H1 拮抗剂

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产品目录号: A10091

库存状态:中国现货中国现货

产品名 目录号 价格 数量
Asenapine maleate 25mg A10091-25
¥ 800.00
Asenapine maleate 50mg A10091-50
¥ 1,000.00
Asenapine maleate 100mg A10091-100
¥ 1,500.00
Asenapine maleate 200mg A10091-200
¥ 2,500.00
Asenapine maleate 10mM * 1mL in DMSO A10091-10mM-D
¥ 720.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

Asenapine shows high affinity (pKi) for numerous receptors, including the serotonin 5-HT1A (8.6), 5-HT1B (8.4), 5-HT2A (10.2), 5-HT2B (9.8), 5-HT2C (10.5), 5-HT5A (8.8), 5-HT6 (9.5), and 5-HT7 (9.9) receptors, the adrenergic α1 (8.9), α2A (8.9), α2B (9.5), and α2C (8.9) receptors, the dopamine D1 (8.9), D2 (8.9), D3 (9.4), and D4 (9.0) receptors, and the histamine H1 (9.0) and H2 (8.2) receptors.

Asenapine maleate

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Chemical Information

目录号 A10091
Mechanism of action Antagonist
分子量 401.84
化学分子式 C17H16ClNO.C4H4O4
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 85650-56-2
Synonyms N/A
SMILES code CN1C[C@H]2[C@H](C1)C3=C(C=CC(=C3)Cl)OC4=CC=CC=C24.C(=C\C(=O)O)\C(=O)O
化学名称 trans-5-Chloro-2,3,3a,12b-tetrahydro-2-methyl-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole maleate

生物活性

Description
Asenapine shows high affinity (pKi) for numerous receptors, including the serotonin 5-HT1A (8.6), 5-HT1B (8.4), 5-HT2A (10.2), 5-HT2B (9.8), 5-HT2C (10.5), 5-HT5A (8.8), 5-HT6 (9.5), and 5-HT7 (9.9) receptors, the adrenergic α1 (8.9), α2A (8.9), α2B (9.5), and α2C (8.9) receptors, the dopamine D1 (8.9), D2 (8.9), D3 (9.4), and D4 (9.0) receptors, and the histamine H1 (9.0) and H2 (8.2) receptors.
Targets
Target Value
5-HT2Cpki: 10.46
5-HT2Apki: 10.15
5-HT7pki: 9.94
5-HT2Bpki: 9.75
5-HT6pki: 9.6
α2B-adrenergicreceptorpki: 9.49
D3receptorpki: 9.38
H1receptorpki: 9
D4receptorpki: 8.95
α1A-adrenergicreceptorpki: 8.93
α2C-adrenergicreceptorpki: 8.91
D2LReceptorpki: 8.9
α2A-adrenergicreceptorpki: 8.9
D1receptorpki: 8.85
5-HT5Apki: 8.84
D2SReceptorpki: 8.84
5-HT1Apki: 8.6
5-HT1Bpki: 8.4
H2receptorpki: 8.21

溶解性

Solubility (25°C)* In vitro DMSO 80 mg/mL (199.08 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.89 mL 124.43 mL 248.86mL
0.5 mM 4.98 mL 24.89 mL 49.77 mL
1 mM 2.49 mL 12.44 mL 24.89 mL
5 mM 0.5 mL 2.49 mL 4.98 mL

*The above data is based on the productmolecular weight 401.84. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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