AT7867 2HCl
目录号: A15006
Akt 抑制剂
AT7867 二盐酸盐是一种强效的 ATP-竞争性抑制剂,针对 Akt1/2/3 和 p70S6K/PKA,其 IC50 分别为 32 nM/17 nM/47 nM 和 85 nM/20 nM,除 AGC激酶家族 外几乎没有活性。
Discription | AT7867 dihydrochloride is a potent ATP-competitive inhibitor of Akt1/2/3 and p70S6K/PKA with IC50 of 32 nM/17 nM/47 nM and 85 nM/20 nM, respectively, little activity outside the AGC kinase family. | ||
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目录号 | A15006 |
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分子式 | C20H22Cl3N3 |
分子量 | 410.77 |
CAS号 | 1431697-86-7 |
SMILES | C1CNCCC1(C2=CC=C(C=C2)C3=CNN=C3)C4=CC=C(C=C4)Cl.Cl.Cl |
其他名称 | AT-7867 dihydrochloride, AT 7867 dihydrochloride |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2