Atipamezole HCl
目录号: A13902
α2 adrenergic receptor 拮抗剂
Atipamezole HCl 是一种选择性的 α2-肾上腺素能受体拮抗剂(Ki 值分别为 α2A、α2B、α2C、α1A 和 α1B 受体的 1.1、1.0、0.89、1300 和 6500 nM)。已被证明能穿透大脑。
Discription | Atipamezole HCl is a selective α2-adrenergic receptor antagonist (Ki values are 1.1, 1.0, 0.89, 1300 and 6500 nM for α2A, α2B, α2C, α1A and α1B receptors respectively). Has been shown to be a brain penetrant. | ||
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目录号 | A13902 |
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分子式 | C14H16N2.HCl |
分子量 | 248.8 |
CAS号 | 104075-48-1 |
SMILES | CCC1(CC2=CC=CC=C2C1)C3=CN=CN3.Cl |
其他名称 | Antisedan |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 12 mg/mL (48.24 mM) | |
Water | 21 mg/mL (84.42 mM) | ||
Ethanol | 48 mg/mL (192.96 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 40.19 mL | 200.96 mL | 401.93 mL |
0.5 mM | 8.04 mL | 40.19 mL | 80.39 mL |
1 mM | 4.02 mL | 20.1 mL | 40.19 mL |
5 mM | 0.8 mL | 4.02 mL | 8.04 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2