Gartisertib (VX-803, ATR inhibitor 2)
Gartisertib (VX-803, ATR inhibitor 2) 是一种 ATP竞争性、口服活性、并且选择性的 ATR抑制剂,其 Ki 值小于150 pM。
Gartisertib (VX-803, ATR inhibitor 2) 是一种 ATP竞争性、口服活性、并且选择性的 ATR抑制剂,其 Ki 值小于150 pM。
| Discription | Gartisertib (VX-803, ATR inhibitor 2) is an ATP-competitive, orally active, and selective ATR inhibitor, with a Ki of <150 pM. |
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| 目录号 | A22162 |
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| 分子式 | C25H29F2N9O3 |
| 分子量 | 541.55 |
| CAS号 | 1613191-99-3 |
| SMILES | O=C(C1=C2N=CC(F)=CN2N=C1N)NC3=C(N4CCC(C(N5CCN(C6COC6)CC5)=O)CC4)C(F)=CN=C3 |
| 其他名称 | M4344 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2