Autotaxin-IN-1
目录号: A19164
autotaxin 抑制剂
Autotaxin-IN-1 是一种强效的自噬素抑制剂,具有良好的效力(IC50=2.2 nM)、药代动力学(PK)属性,以及稳健的药代动力学/药效学(PK/PD)关系。Autotaxin-IN-1 用于治疗骨关节炎疼痛。
Discription | Autotaxin-IN-1 is a potent autotaxin inhibitor, which has favorable potency (IC50=2.2 nM), PK properties, and a robust PK/PD relationship. Autotaxin-IN-1 is used in treatment of osteoarthritis pain. | ||
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目录号 | A19164 |
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分子式 | C21H23N7O2 |
分子量 | 405.45 |
CAS号 | 1619971-30-0 |
SMILES | O=C(N1CC2=NC(NC3CC4=C(C=CC=C4)C3)=NC=C2C1)COCCC5=CN=NN5 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2