Avasimibe (CI-1011)

目录号: A10102

CYP17 抑制剂

Avasimibe (CI-1011)

Avasimibe (CI-1011) Chemical Structure

CAS NO. 166518-60-1

Avasimibe (CI-1011)是口服可生物利用的酰基辅酶A:胆固醇O-酰基转移酶(ACAT)抑制剂,IC50分别为2.9 μM, 13.9 μM和26.5 μM。

库存: 现货

规格 价格 数量
10 mg
¥ 500.00
50 mg
¥ 1,800.00
100 mg
¥ 3,200.00
200 mg
¥ 5,200.00
10mM * 1mL in DMSO
¥ 840.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

Avasimibe (CI-1011)是口服可生物利用的酰基辅酶A:胆固醇O-酰基转移酶(ACAT)抑制剂,IC50分别为2.9 μM, 13.9 μM和26.5 μM。
靶点信息
CYP2C9 ACAT CYP1A2 CYP2C19
2.9 μM3.3 μM13.9 μM26.5 μM
In vitro (25°C) DMSO 100 mg/mL (199.31 mM
Water <1 mg/mL (<1 mM)
Ethanol 8 mg/mL (15.94 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.93 mL 99.66 mL 199.32 mL
0.5 mM 3.99 mL 19.93 mL 39.86 mL
1 mM 1.99 mL 9.97 mL 19.93 mL
5 mM 0.4 mL 1.99 mL 3.99 mL

*The above data is based on the productmolecular weight 501.7 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A10102
作用机制 Inhibitor (抑制剂)
M. Wt 501.7
Formula C29H43NO4S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 166518-60-1
Synonyms CI-1011, CI1011, PD 148515
SMILES CC(C)C1=C(C(=CC=C1)C(C)C)OS(=O)(=O)NC(=O)CC2=C(C=C(C=C2C(C)C)C(C)C)C(C)C

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