Trusted by 10,000+ Scientists since 2006




0 Customer Reviews
产品目录号: A10103


产品名 目录号 价格 数量
Axitinib 50mg A10103-50
¥ 400.00
Axitinib 100mg A10103-100
¥ 700.00
Axitinib 250mg A10103-250
¥ 1,200.00
Axitinib 10mM * 1mL in DMSO A10103-10mM-D
¥ 620.00



Axitinib is a small molecule tyrosine kinase inhibitor,which inhibits multiple targets, including VEGFR-1, VEGFR-2, VEGFR-3, platelet derived growth factor receptor (PDGFR), and cKIT (CD117).





顾客使用 Adooq 产品发表的高质量科研文献
Adooq 顾客使用 Axitinib 发表的文献 (1)
  • Youcef M. Rustum, .et al. Non-Coding Micro RNAs and Hypoxia-Inducible Factors Are Selenium Targets for Development of a Mechanism-Based Combination Strategy in Clear-Cell Renal Cell Carcinoma〞Bench-to-Bedside Therapy, Int J Mol Sci, 2018, Nov; 19(11): 3378 PMID: 30380599

Chemical Information

目录号 A10103
Mechanism of action Inhibitor
分子量 386.5
化学分子式 C22H18N4OS
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 319460-85-0
Synonyms AG 013736
SMILES code CNC(=O)C1=CC=CC=C1SC2=CC3=C(C=C2)C(=NN3)/C=C/C4=CC=CC=N4
化学名称 N-Methyl-2-[[3-[(E)-2-pyridin-2-ylethenyl]-1H-indazol-6-yl]sulfanyl]benzamide


Axitinib is a small molecule tyrosine kinase inhibitor,which inhibits multiple targets, including VEGFR-1, VEGFR-2, VEGFR-3, platelet derived growth factor receptor (PDGFR), and cKIT (CD117).
Target Value
VEGFR1/FLT1IC50: 0.1nM
VEGFR2/Flk1IC50: 0.18nM
VEGFR3IC50: 0.1nM-0.3nM
PDGFRβIC50: 1.6nM
KitIC50: 1.7nM
PDGFRαIC50: 5.0nM
CSF-1RIC50: 73nM
FLT3IC50: >1μM


Solubility (25°C) * In vitro DMSO 35 mg/mL heating (90.56 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 0.5% CMC 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.


Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.87 mL 129.37 mL 258.73mL
0.5 mM 5.17 mL 25.87 mL 51.75 mL
1 mM 2.59 mL 12.94 mL 25.87 mL
5 mM 0.52 mL 2.59 mL 5.17 mL

*The above data is based on the productmolecular weight 386.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Ordering online

To place an order online, simply browse to the product you are interested in and click on the 'Add to Cart' button. To complete this process, you will need to confirm the size and quantity of the products that you require.

To complete an order you will need to register using our simple online registration process. We do not share your contact details with any third parties.

When you are ready to check out simply enter your PO number to complete the ordering process. Please ensure that you send us a copy of your PO by fax or email afterwards.  We will then liaise with you or your purchasing department to confirm the order.

Found your products but not ready to order?

Why not use our WishList feature to store lists of products? This convenient feature allows you to manage lists, append notes to products and share lists with co-workers or colleagues.

Ordering offline

You can email or fax us your purchase order and we will place the order for you. You can also phone us to place the order.  Our contact details are:

We require the following information to process your order:
  • The catalog number for each product. 
  • Your email address or fax number. 
  • Your name and telephone number. 
  • Shipping address and billing address.
  • Purchase order numbers.



Similar product(s)

Keywords:购买 Axitinib | Axitinib 供应商 | 订购 Axitinib | Axitinib 价格 | Axitinib 生产商 | 订单 Axitinib | Axitinib 代理商 | 购买 319460-85-0| 319460-85-0 供应商 | 订购 319460-85-0 | 319460-85-0 价格 | 319460-85-0 生产商 | 订单 319460-85-0 | 319460-85-0 代理商|buy Axitinib | Axitinib Supplier | purchase Axitinib | Axitinib cost | Axitinib manufacturer | order Axitinib | Axitinib distributor | buy 319460-85-0| 319460-85-0 Supplier | purchase 319460-85-0 | 319460-85-0 cost | 319460-85-0 manufacturer | order 319460-85-0 | 319460-85-0 distributor