AZ191

目录号: A14314

DYRK inhibitor

AZ191

AZ191 Chemical Structure

CAS NO. 1594092-37-1

AZ191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM, about 5- and 110-fold selectivity over DYRK1A and DYRK2.

库存: 现货

规格 价格 数量
10 mg
¥ 900.00
25 mg
¥ 1,800.00
50 mg
¥ 2,500.00
10mM * 1mL in DMSO
¥ 660.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

AZ191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM, about 5- and 110-fold selectivity over DYRK1A and DYRK2.
Targets
Dyrk1B (Cell-free assay) DYRK1A (Cell-free assay) DYRK2 (Cell-free assay)
17 nM88 nM1890 nM
In vitro DMSO 86 mg/mL (200.22 mM)
Water <1 mg/mL (<1 mM)
Ethanol 1 mg/mL (2.32 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.28 mL 116.41 mL 232.82 mL
0.5 mM 4.66 mL 23.28 mL 46.56 mL
1 mM 2.33 mL 11.64 mL 23.28 mL
5 mM 0.47 mL 2.33 mL 4.66 mL

*The above data is based on the productmolecular weight 429.52. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

目录号 A14314
MECHANISM OF ACTION Inhibitor
M. Wt 429.52
Formula C24H27N7O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1594092-37-1
Synonyms AZ 191, AZ-191
SMILES CN1CCN(CC1)C2=CC(=C(C=C2)NC3=NC=CC(=N3)C4=CN(C5=C4C=CN=C5)C)OC

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