Azasetron HCl
目录号: A16417
5-HT3 receptor 拮抗剂
Azasetron HCl 是一种选择性的 5-HT3 受体拮抗剂,其 IC50 为 0.33 nM,用于管理由癌症化疗引起的恶心和呕吐。
Discription | Azasetron HCl is a selective 5-HT3 receptor antagonist with IC50 of 0.33 nM used in the management of nausea and vomiting induced by cancer chemotherapy. | ||
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目录号 | A16417 |
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分子式 | C17H20ClN3O3.HCl |
分子量 | 386.27 |
CAS号 | 123040-16-4 |
SMILES | CN1C(=O)COC2=C1C=C(C=C2C(=O)NC3CN4CCC3CC4)Cl.Cl |
其他名称 | Y-25130 hydrochloride, Y25130 hydrochloride, Y 25130 hydrochloride |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | Insoluble | |
Water | 3 mg/mL (7.76 mM) | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 25.89 mL | 129.44 mL | 258.89 mL |
0.5 mM | 5.18 mL | 25.89 mL | 51.78 mL |
1 mM | 2.59 mL | 12.94 mL | 25.89 mL |
5 mM | 0.52 mL | 2.59 mL | 5.18 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2