|Chk1 (Cell-free assay)||Chk2 (Cell-free assay)|
|5 nM||<10 nM|
|In vitro||DMSO||50 mg/mL (137.96 mM)|
|Water||<1 mg/mL (<1 mM)|
|Ethanol||<1 mg/mL (<1 mM)|
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|0.1 mM||27.59 mL||137.97 mL||275.94 mL|
|0.5 mM||5.52 mL||27.59 mL||55.19 mL|
|1 mM||2.76 mL||13.8 mL||27.59 mL|
|5 mM||0.55 mL||2.76 mL||5.52 mL|
*The above data is based on the productmolecular weight 362.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|MECHANISM OF ACTION||Inhibitor|
|Storage||at -20°C 3 years Powder|
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