|0.4 nM||7 nM|
|In vitro (25°C)||DMSO||92 mg/mL (199.46 mM)|
|Water||<1 mg/mL (<1 mM)|
|Ethanol||92 mg/mL (199.46 mM)|
|In vivo||0.5% hydroxyethyl cellulose/0.1% Tween 80||30 mg/mL|
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|0.1 mM||21.68 mL||108.41 mL||216.83 mL|
|0.5 mM||4.34 mL||21.68 mL||43.37 mL|
|1 mM||2.17 mL||10.84 mL||21.68 mL|
|5 mM||0.43 mL||2.17 mL||4.34 mL|
*The above data is based on the productmolecular weight 461.2 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|MECHANISM OF ACTION||Inhibitor|
|Storage||at -20°C 3 years Powder|
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