AZD9496 maleate
目录号: A21726
estrogen receptor (ERα) 拮抗剂
AZD9496 maleate 是一种强效且选择性的雌激素受体(ERα)拮抗剂,IC50 为 0.28 nM。AZD9496 maleate 是一种口服生物利用度高的选择性雌激素受体降解剂(SERD)。
Discription | AZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). |
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目录号 | A21726 |
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分子式 | C29H29F3N2O6 |
分子量 | 558.55 |
CAS号 | 1639042-28-6 |
SMILES | O=C(O)/C=C/C1=CC(F)=C([C@H]2N(CC(C)(F)C)[C@H](C)CC3=C2NC4=C3C=CC=C4)C(F)=C1.O=C(O)/C=C\C(O)=O |
其他名称 | AZD 9496, AZD-9496 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2