BAY-299
目录号: A20239
BRPF2 bromodomain 抑制剂
BAY-299 是一种非常有效的双重抑制剂,其半抑制浓度(IC50)分别为 BRPF2 溴结构域(BD) 67 nM、TAF1 BD2 8 nM 和 TAF1L BD2 106 nM。
Discription | BAY-299 is a very potent, dual inhibitor with IC50s of 67 nM for BRPF2 bromodomains (BD), 8 nM for TAF1 BD2, and 106 nM for TAF1L BD2. | |||||
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Targets |
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Cell Research |
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目录号 | A20239 |
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分子式 | C25H23N3O4 |
分子量 | 429.47 |
CAS号 | 2080306-23-4 |
SMILES | O=C(N1C2=C(C)C=C(N(C)C3=O)C(N3C)=C2)C4=CC=C(CCCO)C5=C4C(C1=O)=CC=C5 |
其他名称 | BAY 299; BAY299 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2