Bay 59-3074
目录号: A16328
CB1/CB2 receptor 激动剂
Bay 59-3074 是一种新型、选择性的 CB1/CB2 受体部分激动剂,其在人类 CB1 和 CB2 受体上的 Ki 值分别为 48.3 和 45.5 nM。
Discription | Bay 59-3074 is a novel, selective CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively . | ||
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Targets |
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目录号 | A16328 |
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分子式 | C18H13F6NO4S |
分子量 | 453.4 |
CAS号 | 406205-74-1 |
SMILES | O=S(OC1=CC(OC2=CC=CC(C(F)(F)F)=C2C#N)=CC=C1)(CCCC(F)(F)F)=O |
其他名称 | Bay59-3074, Bay-59-3074 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 86 mg/mL (189.69 mM) | |
Water | Insoluble | ||
Ethanol | 86 mg/mL (189.69 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 22.06 mL | 110.28 mL | 220.56 mL |
0.5 mM | 4.41 mL | 22.06 mL | 44.11 mL |
1 mM | 2.21 mL | 11.03 mL | 22.06 mL |
5 mM | 0.44 mL | 2.21 mL | 4.41 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2