BC-1215
目录号: A18605
FBXO3 抑制剂
BC-1215 是 F-box 蛋白 3(FBXO3,一种泛素 E3 连接酶组分,IC50=0.9 μg/mL 对 IL-1β释放)的抑制剂。BC-1215 减少 Fbxo3-Fbxl2 之间的相互作用,并阻止 SCFFbxo3 催化的 Fbxl2 泛素化。
Discription | BC-1215 is an inhibitor of F-box protein 3 (FBXO3, a ubiquitin E3 ligase component, IC50=0.9 μg/mL for IL-1β release). BC-1215 decreases Fbxo3-Fbxl2 interaction and prevents SCFFbxo3 catalyzed Fbxl2 ubiquitination. |
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目录号 | A18605 |
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分子式 | C26H26N4 |
分子量 | 394.51 |
CAS号 | 1507370-20-8 |
SMILES | C1(CNCCNCC2=CC=C(C3=NC=CC=C3)C=C2)=CC=C(C4=NC=CC=C4)C=C1 |
其他名称 | BC1215, BC 1215 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2