BGB-102
目录号: A21288
EGFR/HER2/HER4 抑制剂
BGB-102 是一种强效的多激酶抑制剂,针对 EGFR、HER2 和 HER4,其半抑制浓度(IC50)分别为 9.6 nM、18 nM 和 40.3 nM。
EGFR/HER2/HER4 抑制剂
Discription | BGB-102 is a potent multi-kinase inhibitor against EGFR, HER2, and HER4 with IC50s of 9.6 nM, 18 nM and 40.3 nM, respectively. |
---|
目录号 | A21288 |
---|---|
分子式 | C22H25BrN4O2 |
分子量 | 457.36 |
CAS号 | 807640-87-5 |
SMILES | CN1CCCCCOC(C(OC)=C2)=CC3=C2N=CN/C3=N\C4=CC(Br)=CC=C4C1 |
其他名称 | JNJ-26483327 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2