BI-3812
目录号: A20311
BCL6 抑制剂
BI-3812 是一种强效且有效的 BCL6 抑制剂,它抑制 BCL6 的 BTB 域,具有约3纳摩尔的 IC50;BI-3812 具有抗肿瘤活性。
Discription | BI-3812 is potent and efficacious BCL6 inhibitor, inhibiting the BTB domain of BCL6, with an IC50 of ??3 nM; BI-3812 has antitumor activity. |
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目录号 | A20311 |
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分子式 | C26H32ClN7O5 |
分子量 | 558.03 |
CAS号 | 2166387-64-8 |
SMILES | ClC1=CN=C(N2CCC(C(N(C)C)=O)CC2)N=C1NC3=CC(C=C(OCC(NC)=O)C(N4C)=O)=C4C(OC)=C3 |
其他名称 | BI3812, BI 3812 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 12 mg/mL (21.5 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 17.92 mL | 89.6 mL | 179.2 mL |
0.5 mM | 3.58 mL | 17.92 mL | 35.84 mL |
1 mM | 1.79 mL | 8.96 mL | 17.92 mL |
5 mM | 0.36 mL | 1.79 mL | 3.58 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2