BI-D1870 Chemical Structure

CAS NO. 501437-28-1

BI-D1870 is a potent and specific inhibitor of the p90 ribosomal S6 kinase (RSK) isoforms in vitro and in vivo, which inhibits RSK1, RSK2, RSK3 and RSK4 in vitro with an IC50 of 10–30 nM.

库存: 现货

规格 价格 数量
5 mg
¥ 1,100.00
10 mg
¥ 1,900.00
25 mg
¥ 3,400.00
50 mg
¥ 5,300.00
10mM * 1mL in DMSO
¥ 1,100.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

BI-D1870 is a potent and specific inhibitor of the p90 ribosomal S6 kinase (RSK) isoforms in vitro and in vivo, which inhibits RSK1, RSK2, RSK3 and RSK4 in vitro with an IC50 of 10–30 nM.
靶点信息
RSK4 (Cell-free assay) RSK3 (Cell-free assay) RSK2 (Cell-free assay) RSK1 (Cell-free assay)
15 nM18 nM24 nM31 nM
In vitro (25°C) DMSO 78 mg/mL (199.27 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% PEG400/0.5% Tween80/5% propylene glycol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.55 mL 127.74 mL 255.49 mL
0.5 mM 5.11 mL 25.55 mL 51.1 mL
1 mM 2.55 mL 12.77 mL 25.55 mL
5 mM 0.51 mL 2.55 mL 5.11 mL

*The above data is based on the productmolecular weight 391.41. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A12452
MECHANISM OF ACTION Inhibitor
M. Wt 391.41
Formula C19H23F2N5O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 501437-28-1
Synonyms N/A
SMILES CC1C(=O)N(C2=CN=C(N=C2N1CCC(C)C)NC3=CC(=C(C(=C3)F)O)F)C

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