BKI-1369
目录号: A18678
bumped kinase 抑制剂
BKI-1369 是一种凸起激酶抑制剂(BKI)。BKI-1369 增强了人类Ether-a-go-go相关基因(hERG)的抑制活性,其半抑制浓度(IC50)为1.52微摩尔。
Discription | BKI-1369 is a bumped kinase inhibitor (BKI). BKI-1369 increases human Ether-a-go-go-related gene (hERG)-inhibitory activity with an IC50 of 1.52 μM. | |||||
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Cell Research |
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目录号 | A18678 |
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分子式 | C23H27N7O |
分子量 | 417.51 |
CAS号 | 1951431-22-3 |
SMILES | NC1=C2C(N(CC3CCN(C)CC3)N=C2C4=CC=C5N=C(OCC)C=CC5=C4)=NC=N1 |
其他名称 | BKI1369, BKI 1369 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2