|3 nM||150 nM||493 nM||591 nM|
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|0.1 mM||19.63 mL||98.16 mL||196.32 mL|
|0.5 mM||3.93 mL||19.63 mL||39.26 mL|
|1 mM||1.96 mL||9.82 mL||19.63 mL|
|5 mM||0.39 mL||1.96 mL||3.93 mL|
*The above data is based on the productmolecular weight 509.38. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|MECHANISM OF ACTION||Inhibitor|
|Storage||at -20°C 3 years Powder|
|Synonyms||BLU-9931, BLU 9931|
BGJ398 is a potent and selective inhibitor with potential antiangiogenic and antineoplastic activities of fibroblast growth factor receptor…
NVP-BGJ398 phosphate is a novel selective, pan-specific FGFR inhibitor with IC50 of 0.9, 1.4, and 1 nM for FGFR1, FGFR2, and FGFR3, respect…
PD173074 is a potent, cell permeable and ATP competitive inhibitor of FGFR and VEGFR.
Debio-1347 is an orally bioavailable inhibitor of the fibroblast growth factor receptor subtypes 1 (FGFR-1), 2 (FGFR-2) and 3 (FGFR-3), with…
Alofanib is a potent and selective allosteric inhibitor of FGFR2 with potential anticancer activity.
Pazopanib is a potent and selective multi-targeted receptor tyrosine kinase inhibitor of VEGFR-1, VEGFR-2, VEGFR-3, PDGFR-a/β, and c-kit th…