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BMY 7378是5-HT1A部分激动剂和高亲和力α1D肾上腺素能受体拮抗剂。
Targets
| Target | Value |
|---|---|
| 5-HT1A | pIC50: 8.3 |
| α1D-adrenoceptor | pki: 8.2 |
| DopamineD2receptor | pIC50: 7.4 |
| α2C-adrenoceptor | pki: 6.54 |
| 5-HT1C | pIC50: 6.4 |
| 5-HT1D | pIC50: 5.9 |
| H1receptor | pIC50: 5.7 |
| 5-HT2 | pIC50: 5.5 |
| H2receptor | pIC50: 5.3 |
| α2-adrenoceptor | pIC50: 5.1 |
| β1-adrenoceptor | pIC50: 5.1 |
| DopamineD1receptor | pIC50: 5 |
| Nicotinicreceptor | pIC50: 4.9 |
| β2-adrenoceptor | pIC50: <5.0 |
| 5-HT3 | pIC50: <5.0 |
| H3receptor | pIC50: <5.0 |
| GABAAreceptor | pIC50: <5.0 |
| GABABreceptor | pIC50: <5.0 |
| MuscarinicM1receptor | pIC50: <5.0 |
| MuscarinicM2receptor | pIC50: <5.0 |
| MuscarinicM3receptor | pIC50: <5.0 |
| NMDAreceptor | pIC50: <5.0 |
| AT1receptor | pIC50: <5.0 |
| AT2receptor | pIC50: <5.0 |
| EndothelinReceptor | pIC50: <5.0 |
| AdenosineA1receptor | pIC50: <5.0 |
| AdenosineA2receptor | pIC50: <5.0 |
| In vitro (25°C) | DMSO | 81 mg/mL (176.69 mM) | |
| Water | 81 mg/mL (176.69 mM) | ||
| Ethanol | 18 mg/mL (39.26 mM) | ||
| In vivo | Saline | 14 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 21.81 mL | 109.07 mL | 218.14 mL |
| 0.5 mM | 4.36 mL | 21.81 mL | 43.63 mL |
| 1 mM | 2.18 mL | 10.91 mL | 21.81 mL |
| 5 mM | 0.44 mL | 2.18 mL | 4.36 mL |
*The above data is based on the productmolecular weight 458.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| 目录号 | A11208 |
|---|---|
| 作用机制 | Agonist (激动剂) |
| M. Wt | 458.42 |
| Formula | C22H31N3O3.2HCl |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
| CAS No. | 21102-95-4 |
| Synonyms | BMY7378, BMY-7378 |
| SMILES | COC1=CC=CC=C1N2CCN(CC2)CCN3C(=O)CC4(CCCC4)CC3=O.Cl.Cl |
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