Trusted by 10,000+ Scientists since 2006
微信关注
申请试用装

BRL-15572

5-HT1D receptor 拮抗剂

0 Customer Reviews
产品目录号: A11178

库存状态:中国现货中国现货

产品名 目录号 价格 数量
BRL-15572 5mg A11178-5
¥ 500.00
BRL-15572 10mg A11178-10
¥ 700.00
BRL-15572 50mg A11178-50
¥ 2,600.00
BRL-15572 100mg A11178-100
¥ 4,200.00
BRL-15572 10mM * 1mL in DMSO A11178-10mM-D
¥ 1,030.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

BRL-15572 is a selective h5-HT1D antagonist, displaying 60-fold selectivity over h5-HT1B, and exhibiting little or no affinity for a range of other receptor types.

BRL-15572

双击上述图片即可查看完整大小

缩小
放大

更多视图

顾客使用 Adooq 产品发表的高质量科研文献

Chemical Information

目录号 A11178
Mechanism of action Antagonist
分子量 443.42
化学分子式 C25H27ClN2O.HCl
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 193611-72-2
Synonyms BRL15572
SMILES code C1CN(CCN1CC(C(C2=CC=CC=C2)C3=CC=CC=C3)O)C4=CC(=CC=C4)Cl.Cl.Cl
化学名称 3-[4-(4-Chlorophenyl)piperazin-1-yl ]-1,1-diphenyl-2-propanol hydrochloride

生物活性

Description

BRL-15572 is a selective h5-HT1D antagonist, displaying 60-fold selectivity over h5-HT1B, and exhibiting little or no affinity for a range of other receptor types.

Targets
Target Value
5-HT1Dpki: 7.9
5-HT1Apki: 7.7
5-HT2Bpki: 7.4
5-HT2Apki: 6.6
5-HT7pki: 6.3
5-HT2Cpki: 6.2
5-HT1Bpki: 6.1
5-HT1Fpki: 6
5-HT6pki: 5.9
5-HT1Epki: 5.2

溶解性

Solubility (25°C) * In vitro DMSO 96 mg/mL (200.05 mM)
Water <1 mg/mL (<1 mM)
Ethanol 40 mg/mL (83.35 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 20 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.55 mL 112.76 mL 225.52mL
0.5 mM 4.51 mL 22.55 mL 45.1 mL
1 mM 2.26 mL 11.28 mL 22.55 mL
5 mM 0.45 mL 2.26 mL 4.51 mL

*The above data is based on the productmolecular weight 443.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Ordering online

To place an order online, simply browse to the product you are interested in and click on the 'Add to Cart' button. To complete this process, you will need to confirm the size and quantity of the products that you require.

To complete an order you will need to register using our simple online registration process. We do not share your contact details with any third parties.

When you are ready to check out simply enter your PO number to complete the ordering process. Please ensure that you send us a copy of your PO by fax or email afterwards.  We will then liaise with you or your purchasing department to confirm the order.

Found your products but not ready to order?

Why not use our WishList feature to store lists of products? This convenient feature allows you to manage lists, append notes to products and share lists with co-workers or colleagues.

Ordering offline

You can email or fax us your purchase order and we will place the order for you. You can also phone us to place the order.  Our contact details are:

We require the following information to process your order:
  • The catalog number for each product. 
  • Your email address or fax number. 
  • Your name and telephone number. 
  • Shipping address and billing address.
  • Purchase order numbers.

产品标签

使用空格分隔标签。使用单引号(')标注词组。


Keywords:购买 BRL-15572 | BRL-15572 供应商 | 订购 BRL-15572 | BRL-15572 价格 | BRL-15572 生产商 | 订单 BRL-15572 | BRL-15572 代理商 | 购买 193611-72-2| 193611-72-2 供应商 | 订购 193611-72-2 | 193611-72-2 价格 | 193611-72-2 生产商 | 订单 193611-72-2 | 193611-72-2 代理商|buy BRL-15572 | BRL-15572 Supplier | purchase BRL-15572 | BRL-15572 cost | BRL-15572 manufacturer | order BRL-15572 | BRL-15572 distributor | buy 193611-72-2| 193611-72-2 Supplier | purchase 193611-72-2 | 193611-72-2 cost | 193611-72-2 manufacturer | order 193611-72-2 | 193611-72-2 distributor