BRL-54443

Name: BRL-54443
SKU: A15592

目录号: A15592

5-HT1E/5-HT1F receptor 激动剂

BRL-54443 Chemical Structure

CAS NO. 57477-39-1

BRL 54443是5-HT1E和5-HT1F受体激动剂，pKi分别为8.7和9.25，对5-HT1A，5-HT1B，5-HT1D受体的结合亲和力较弱。

库存：现货

规格	价格	数量
10 mg	￥ 700.00
25 mg	￥ 1,400.00
100 mg	￥ 5,500.00

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生物活性

BRL 54443是5-HT1E和5-HT1F受体激动剂，pKi分别为8.7和9.25，对5-HT1A，5-HT1B，5-HT1D受体的结合亲和力较弱。

溶解度 *

In vitro (25°C)	DMSO	40 mg/mL (173.68 mM)
	Water	Insoluble
	Ethanol	2 mg/mL (8.68 mM)
In vivo	30% propylene glycol, 5% Tween 80, 65% D5W	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	43.42 mL	217.1 mL	434.2 mL
0.5 mM	8.68 mL	43.42 mL	86.84 mL
1 mM	4.34 mL	21.71 mL	43.42 mL
5 mM	0.87 mL	4.34 mL	8.68 mL

*The above data is based on the productmolecular weight 230.31. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15592
作用机制	Agonist (激动剂)
M. Wt	230.31
Formula	C14H18N2O
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	57477-39-1
Synonyms	BRL54443, BRL 54443
SMILES	CN1CCC(CC1)C2=CNC3=C2C=C(C=C3)O