Bromocriptin mesylate
目录号: A13705
dopamine D2 receptor 激动剂
溴隐亭甲磺酸盐是一种强效的多巴胺受体激动剂,它与D2受体具有最高亲和力(Ki = 2.5 nM)。因此,它已被用于帕金森病的联合治疗中。
Discription | Bromocriptine mesylate is a potent dopamine receptor agonist that binds the D2 receptor with highest affinity (Ki = 2.5 nM).1,2 As a result, it has found applications in combination therapy for Parkinsonism. | |||||
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Cell Research |
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目录号 | A13705 |
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分子式 | C32H40BrN5O5.CH3SO3H |
分子量 | 750.7 |
CAS号 | 22260-51-1 |
SMILES | CC(C)C[C@H]1C(=O)N2CCC[C@H]2[C@]3(N1C(=O)[C@](O3)(C(C)C)NC(=O)[C@H]4CN([C@@H]5CC6=C(NC7=CC=CC(=C67)C5=C4)Br)C)O.CS(=O)(=O)O |
其他名称 | CB 154, Parlodel, Cycloset |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2