BX-912

目录号: A11149

PDK1 抑制剂

BX-912

BX-912 Chemical Structure

CAS NO. 702674-56-4

BX-912是3-磷酸肌醇依赖性激酶1(PDK1)的抑制剂。

库存: 现货

规格 价格 数量
5 mg
¥ 900.00
10 mg
¥ 1,600.00
50 mg
¥ 5,200.00
100 mg
¥ 7,800.00
10mM * 1mL in DMSO
¥ 1,440.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

BX-912是3-磷酸肌醇依赖性激酶1(PDK1)的抑制剂。
Targets
Target Value
PDK-1IC50: 12nM
PKAIC50: 110nM
KDRIC50: 410nM
CDK2/CyclinEIC50: 650nM
Chk1IC50: 830nM
c-KitIC50: 850nM
PKCIC50: 1.25μM
T-FynIC50: 2.1μM
Insulin ReceptorIC50: 6.1μM
GSK-3βIC50: 7.4μM
EGFRIC50: >10μM
In vitro (25°C) DMSO 80 mg/mL (169.72 mM)
Water Insoluble
Ethanol 80 mg/mL (169.72 mM)
In vivo 30% PEG400+0.5% Tween80+5% propylene glycol 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.21 mL 106.07 mL 212.13 mL
0.5 mM 4.24 mL 21.21 mL 42.43 mL
1 mM 2.12 mL 10.61 mL 21.21 mL
5 mM 0.42 mL 2.12 mL 4.24 mL

*The above data is based on the productmolecular weight 471.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11149
作用机制 Inhibitor (抑制剂)
M. Wt 471.4
Formula C20H23BrN8O
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 702674-56-4
Synonyms BX912
SMILES C1CCN(C1)C(=O)NC2=CC=CC(=C2)NC3=NC=C(C(=N3)NCCC4=CN=CN4)Br

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