Cariprazine
目录号: A21202
D3 receptor and D2 receptor partial 激动剂
Cariprazine 是一种新型抗精神病药物候选物,对 D3 受体(Ki=0.085 nM)和 D2 受体(Ki=0.49 nM)表现出高亲和力,对 5-HT1A 受体(Ki=2.6 nM)则表现出中等亲和力。
Discription | Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). | |||||
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Cell Research |
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目录号 | A21202 |
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分子式 | C21H32Cl2N4O |
分子量 | 427.41 |
CAS号 | 839712-12-8 |
SMILES | O=C(N[C@H]1CC[C@H](CCN2CCN(C3=CC=CC(Cl)=C3Cl)CC2)CC1)N(C)C |
其他名称 | RGH-188, RGH 188, RGH188 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2