RS-127445
RS-127445 是一种强效且选择性的5-HT2B受体拮抗剂，其对于与之密切相关的5-HT2A和5-HT2C受体的选择性约为1000倍。
顾客使用 Adooq 产品发表的高质量科研文献
Adooq用户使用RS-127445发表的1篇文献
生物活性
| Discription | RS-127445 is a potent and selective antagonist at the serotonin 5-HT2B receptor, with around 1000x selectivity over the closely related 5-HT2A and 5-HT2C receptors. |
|||||
|---|---|---|---|---|---|---|
| Targets |
|
|||||
| Cell Research |
|
产品信息
| 目录号 | A11165 |
|---|---|
| 分子式 | C17H16FN3 |
| 分子量 | 281.33 |
| CAS号 | 199864-87-4 |
| SMILES | CC(C)C1=NC(=NC(=C1)C2=CC=C(C3=CC=CC=C32)F)N |
| 其他名称 | RS127445, MT 500, RS127,445 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro | DMSO | 54 mg/mL (191.94 mM) | |
| Water | Insoluble | ||
| Ethanol | 8 mg/mL (28.43 mM) | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 35.55 mL | 177.73 mL | 355.45 mL |
| 0.5 mM | 7.11 mL | 35.55 mL | 71.09 mL |
| 1 mM | 3.55 mL | 17.77 mL | 35.55 mL |
| 5 mM | 0.71 mL | 3.55 mL | 7.11 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
Keywords: 购买 RS-127445 | RS-127445 供应商 | RS-127445 花费 | RS-127445 生产商 | 订购 RS-127445 | RS-127445 代理商
| 购买 199864-87-4 | 199864-87-4 供应商 | 199864-87-4 花费 | 199864-87-4 生产商 | 订购 199864-87-4 | 199864-87-4 代理商