Limantrafin (CB-103)
目录号: A22160
Notch 抑制剂
CB-103 是一种首创的、口服活性的蛋白-蛋白相互作用(PPI)抑制剂,针对的是 NOTCH 转录激活复合体。CB-103 具有抗肿瘤活性。
Notch 抑制剂
Discription | CB-103 is a first-in-class, orally active protein-protein interaction (PPI) inhibitor of the NOTCH transcriptional activation complex. CB-103 has anti-tumor activity. |
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目录号 | A22160 |
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分子式 | C15H18N2O |
分子量 | 242.32 |
CAS号 | 218457-67-1 |
SMILES | NC1=CC=C(OC2=CC=C(C(C)(C)C)C=C2)N=C1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2