CB1954
目录号: A15862
CB1954 是一种抗癌前药，它在酶 NQO2 和辅助底物 caricotamide (EP-0152R) (EP) 的存在下转化为一种强效的双功能烷化剂。它可以被 NAD(P)H 醌氧化还原酶 2 激活。
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生物活性
| Discription | CB1954 is a anticancer prodrug that is converted in the presence of the enzyme NQO2 and co-substrate caricotamide ( EP-0152R) (EP) into a potent cytotoxic bifunctional alkylating agent.It can be activated by NAD(P)H quinone oxidoreductase 2. | |||||
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| Cell Research |
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产品信息
| 目录号 | A15862 |
|---|---|
| 分子式 | C9H8N4O5 |
| 分子量 | 252.18 |
| CAS号 | 21919-05-1 |
| SMILES | O=C(N)C1=CC(N2CC2)=C([N+]([O-])=O)C=C1[N+]([O-])=O |
| 其他名称 | Tretazicar |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro | DMSO | 49 mg/mL (194.3 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 39.65 mL | 198.27 mL | 396.54 mL |
| 0.5 mM | 7.93 mL | 39.65 mL | 79.31 mL |
| 1 mM | 3.97 mL | 19.83 mL | 39.65 mL |
| 5 mM | 0.79 mL | 3.97 mL | 7.93 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 21919-05-1 | 21919-05-1 供应商 | 21919-05-1 花费 | 21919-05-1 生产商 | 订购 21919-05-1 | 21919-05-1 代理商