CCT-251921
目录号: A20610
CDK8 抑制剂
CCT-251921 是一种效力强大、选择性高、且可口服的 CDK8 抑制剂,其 IC50 为 2.3 nM。
Discription | CCT-251921 is a potent, selective, and orally bioavailable CDK8 inhibitor with an IC50 of 2.3 nM. | |||||
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Targets |
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Cell Research |
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目录号 | A20610 |
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分子式 | C21H23ClN6O |
分子量 | 410.9 |
CAS号 | 1607837-31-9 |
SMILES | O=C1NCCC12CCN(C3=C(Cl)C(N)=NC=C3C4=CC5=C(N(C)N=C5)C=C4)CC2 |
其他名称 | CCT251921;CCT 251921 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2