CCT128930

目录号: A11031

AKT Inhibitor

CCT128930

CCT128930 Chemical Structure

CAS NO. 885499-61-6

CCT128930 is an ATP-competitive AKT inhibitor that is a potent, advanced lead pyrrolopyrimidine compound exhibiting selectivity for AKT over PKA, achieved by targeting a single amino acid difference.

库存: 现货

规格 价格 数量
10 mg
¥ 1,280.00
25 mg
¥ 2,560.00
50 mg
¥ 4,500.00
100 mg
¥ 7,200.00
10mM * 1mL in DMSO
¥ 1,030.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

CCT128930 is an ATP-competitive AKT inhibitor that is a potent, advanced lead pyrrolopyrimidine compound exhibiting selectivity for AKT over PKA, achieved by targeting a single amino acid difference.
Targets
Akt2 (Cell-free assay) p70 S6K (Cell-free assay) PKA (Cell-free assay)
6 nM120 nM168 nM
In vitro (25°C) DMSO 68 mg/mL (198.92 mM)
Water <1 mg/mL (<1 mM)
Ethanol 6 mg/mL (17.55 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 11 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.26 mL 146.28 mL 292.57 mL
0.5 mM 5.85 mL 29.26 mL 58.51 mL
1 mM 2.93 mL 14.63 mL 29.26 mL
5 mM 0.59 mL 2.93 mL 5.85 mL

*The above data is based on the productmolecular weight 341.8 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

目录号 A11031
MECHANISM OF ACTION Inhibitor
M. Wt 341.8
Formula C18H20ClN5
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 885499-61-6
Synonyms CCT-128930
SMILES C1CN(CCC1(CC2=CC=C(C=C2)Cl)N)C3=NC=NC4=C3C=CN4

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