CD-161
目录号: A18921
BET 抑制剂
CD-161 是一种效力强大且可口服生物利用的 BET 抑制剂,其 IC50 分别为 BRD4 BD1 的 28.2 nM 和 BRD4 BD2 的 7.2 nM。
Discription | CD-161 is a potent and orally bioavailable BET inhibitor with an IC50s of 28.2 nM and 7.2 nM for BRD4 BD1 and BRD4 BD2, respectively. | |||||
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Cell Research |
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目录号 | A18921 |
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分子式 | C26H21N5O2 |
分子量 | 435.48 |
CAS号 | 1627716-22-6 |
SMILES | CC1=C(C2=CC3=C(C=C2OC)C4=C(C5=CC=NC6=CC=CC=C56)N=C(C)N=C4N3)C(C)=NO1 |
其他名称 | CD-161; CD161; CD 161 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2