CDK12-IN-3
目录号: A19768
CDK12 抑制剂
CDK12-IN-3 是一种效力强大且选择性高的 CDK12 抑制剂,在酶学测定中的 IC50 为 491 nM。
Discription | CDK12-IN-3 is a potent and selective CDK12 inhibitor with an IC50 of 491 nM in enzymatic assay. | ||
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Targets |
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目录号 | A19768 |
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分子式 | C23H28F2N8O |
分子量 | 470.52 |
CAS号 | 2220184-50-7 |
SMILES | CC(C)N1C2=NC(N3CCCC[C@H]3CCO)=NC(NCC4=NC5=C(C(F)=C(F)C=C5)N4)=C2N=C1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2