CDK8/19-IN-1
目录号: A19986
CDK8/19 dual 抑制剂
CDK8/19-IN-1 是一种高效、选择性且可口服的 CDK8/19 双重抑制剂,其 IC50 分别为 0.46 nM、0.99 nM 和 270 nM,针对 CDK8、CDK19 和 CDK9。
| Discription | CDK8/19-IN-1 is a potent, selective and oral bioavailable CDK8/19 dual inhibitor, with IC50s of 0.46 nM, 0.99 nM and 270 nM for CDK8, CDK19 and CDK9, respectively. | |||||
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| 目录号 | A19986 |
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| 分子式 | C19H18N4O4S2 |
| 分子量 | 430.5 |
| CAS号 | 1818427-07-4 |
| SMILES | O=C(C1=C2CCC3=C(SN=C3)C2=C(OC4=CC=C(C(NCCOC)=O)N=C4)S1)N |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2