CH5132799

目录号: A11169

PI3K inhibitor

CH5132799 Chemical Structure

CAS NO. 1007207-67-1

CH5132799 is a novel class I PI3K inhibitor, which exhibited a strong inhibitory activity especially against PI3Kα (IC(50)=0.014 μM).

库存: 现货

规格 价格 数量
5 mg
¥ 1,800.00
10 mg
¥ 2,800.00
50 mg
¥ 7,800.00
100 mg
¥ 11,000.00
10mM * 1mL in DMSO
¥ 1,950.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

CH5132799 is a novel class I PI3K inhibitor, which exhibited a strong inhibitory activity especially against PI3Kα (IC(50)=0.014 μM).

Targets
Target Value
PI3KαIC50: 14nM
PI3KγIC50: 36nM
PI3KβIC50: 0.12μM
PI3KδIC50: 0.50μM
mTORIC50: 1.6μM
C2βIC50: 5.3μM
C2αIC50: >10μM
Vps34IC50: >10μM
In vitro (25°C) DMSO 12 mg/mL (31.79 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.5 mL 132.48 mL 264.96 mL
0.5 mM 5.3 mL 26.5 mL 52.99 mL
1 mM 2.65 mL 13.25 mL 26.5 mL
5 mM 0.53 mL 2.65 mL 5.3 mL

*The above data is based on the productmolecular weight 377.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11169
MECHANISM OF ACTION Inhibitor
M. Wt 377.42
Formula C15H19N7O3S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1007207-67-1
Synonyms CH-5132799
SMILES CS(=O)(=O)N1CCC2=C(N=C(N=C21)N3CCOCC3)C4=CN=C(N=C4)N

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