CI-1044
目录号: A20492
PDE4 抑制剂
CI-1044 是一种口服活性的 PDE4 抑制剂,其 IC50 分别为 0.29, 0.08, 0.56, 0.09 μM,针对 PDE4A5, PDE4B2, PDE4C2 和 PDE4D3。
Discription | CI-1044 is an orally active PDE4 inhibitor with IC50s of 0.29, 0.08, 0.56, 0.09 μM for PDE4A5, PDE4B2, PDE4C2 and PDE4D3, respectively. | ||
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目录号 | A20492 |
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分子式 | C23H19N5O2 |
分子量 | 397.43 |
CAS号 | 197894-84-1 |
SMILES | O=C(C1=CC=CN=C1)N[C@H]2C(N3C4=C(CC3)C=C(N)C=C4C(C5=CC=CC=C5)=N2)=O |
其他名称 | CI 1044, CI1044; PD-189659, PD189659, PD 189659 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2