CID16020046
目录号: A16818
GPR55 拮抗剂
CID16020046 是一种选择性的 GPR55 拮抗剂,能够抑制酵母中 GPR55 的固有活性,其 IC50 为 0.15 微摩尔。它对其他广泛的 GPCRs、离子通道、激酶和核受体表现出较弱的活性。
Discription | CID16020046 is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast. It demonstrates weak activity against a broad spectrum of other GPCRs, ion channels, kinases, and nuclear receptor. |
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目录号 | A16818 |
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分子式 | C25H19N3O4 |
分子量 | 425.44 |
CAS号 | 834903-43-4 |
SMILES | O=C(O)C1=CC=C(N(C2=O)C(C3=CC=CC(O)=C3)C4=C2NN=C4C5=CC=C(C)C=C5)C=C1 |
其他名称 | C390-0219, CID 16020046, CID-16020046 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 77 mg/mL (180.99 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 23.51 mL | 117.53 mL | 235.05 mL |
0.5 mM | 4.7 mL | 23.51 mL | 47.01 mL |
1 mM | 2.35 mL | 11.75 mL | 23.51 mL |
5 mM | 0.47 mL | 2.35 mL | 4.7 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2