Clemastine fumarate
目录号: A10226
Histamine Receptor antagonis
克莱马斯汀是一种选择性的组胺H1受体拮抗剂。它与组胺H1受体结合,从而阻断了内源性组胺的作用,这导致了由组胺引起的负面症状的暂时缓解。
Discription | Clemastine is a selective histamine H1 antagonist. It binds to the histamine H1 receptor, thus blocking the action of endogenous histamine, which leads to temporary relief of the negative symptoms caused by histamine. | ||
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目录号 | A10226 |
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分子式 | C21H26ClNO.C4H4O4 |
分子量 | 459.96 |
CAS号 | 14976-57-9 |
SMILES | C[C@@](C1=CC=CC=C1)(C2=CC=C(C=C2)Cl)OCC[C@H]3CCCN3C.C(=C/C(=O)O)\C(=O)O |
其他名称 | meclastin |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | Warmed: 31 mg/mL (67.39 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 21.74 mL | 108.71 mL | 217.41 mL |
0.5 mM | 4.35 mL | 21.74 mL | 43.48 mL |
1 mM | 2.17 mL | 10.87 mL | 21.74 mL |
5 mM | 0.43 mL | 2.17 mL | 4.35 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2