CPI-169

目录号: A15920

EZH2 抑制剂

CPI-169

CPI-169 Chemical Structure

CAS NO. 1450655-76-1

CPI-169是一种有效的选择性EZH2抑制剂,对EZH2 WT,EZH2 Y641N和EZH1的IC50分别为0.24 nM,0.51 nM和6.1 nM。

库存: 现货

规格 价格 数量
5 mg
¥ 1,200.00
10 mg
¥ 1,800.00
25 mg
¥ 4,200.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

CPI-169是一种有效的选择性EZH2抑制剂,对EZH2 WT,EZH2 Y641N和EZH1的IC50分别为0.24 nM,0.51 nM和6.1 nM。
靶点信息
EZH2 WT EZH2 Y641N EZH1
0.24 nM0.51 nM6.1 nM
In vitro (25°C) DMSO 88 mg/mL (166.45 mM)
Water Insoluble
Ethanol 88 mg/mL (166.45 mM)
In vivo 10% DMSO+60% PEG 400+30% ddH2O 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.92 mL 94.58 mL 189.16 mL
0.5 mM 3.78 mL 18.92 mL 37.83 mL
1 mM 1.89 mL 9.46 mL 18.92 mL
5 mM 0.38 mL 1.89 mL 3.78 mL

*The above data is based on the productmolecular weight 528.66. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A15920
作用机制 Inhibitor (抑制剂)
M. Wt 528.66
Formula C27H36N4O5S
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 1450655-76-1
Synonyms CPI 169, CPI169
SMILES CCS(N1CCC([C@@](N2C(C)=C(/C(O)=N/CC(C(O)=N3)=C(OC)C=C3C)C4=CC=CC=C42)([H])C)CC1)(=O)=O

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