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BET bromodomain 抑制剂

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产品目录号: A13068


产品名 目录号 价格 数量
CPI-203 5mg A13068-5
¥ 900.00
CPI-203 10mg A13068-10
¥ 1,700.00
CPI-203 25mg A13068-25
¥ 3,500.00
CPI-203 50mg A13068-50
¥ 5,500.00



CPI203 is a novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 with an IC50 of ~37 nM (BRD4 α-screen assay).





顾客使用 Adooq 产品发表的高质量科研文献
Adooq 顾客使用 CPI-203 发表的文献 (1)
  • Derenzini E, .et al. BET Inhibition-Induced GSK3汕 Feedback Enhances Lymphoma Vulnerability to PI3K Inhibitors, Cell Rep, 2018, Aug 21;24(8):2155-2166 PMID: 30134175

Chemical Information

目录号 A13068
Mechanism of action Inhibitor
分子量 399.9
化学分子式 C19H18ClN5OS
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 1446144-04-2
Synonyms 0
SMILES code CC1=C(SC2=C1C(=N[C@H](C3=NN=C(N32)C)CC(=O)N)C4=CC=C(C=C4)Cl)C
化学名称 (S)-2-(4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetamide


CPI203 is a novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 with an IC50 of ~37 nM (BRD4 α-screen assay).


Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.01 mL 125.03 mL 250.06mL
0.5 mM 5 mL 25.01 mL 50.01 mL
1 mM 2.5 mL 12.5 mL 25.01 mL
5 mM 0.5 mL 2.5 mL 5 mL

*The above data is based on the productmolecular weight 399.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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