CPI-268456

Name: CPI-268456
SKU: A15828

目录号: A15828

CPI-268456 Chemical Structure

CAS NO. 1380087-86-4

CPI-268456是含溴结构域蛋白4（BRD4）的配体。它与BRD4结合（无细胞试验中IC50 = <0.5 ?M），并抑制THP-1细胞中LPS诱导的IL-6分泌（IC50 = <0.5 ?M）。

库存：现货

规格	价格	数量
5 mg	￥ 1,400.00
10 mg	￥ 2,500.00
25 mg	￥ 5,500.00

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生物活性

CPI-268456是含溴结构域蛋白4（BRD4）的配体。它与BRD4结合（无细胞试验中IC50 = <0.5 ?M），并抑制THP-1细胞中LPS诱导的IL-6分泌（IC50 = <0.5 ?M）。

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	25.06 mL	125.3 mL	250.6 mL
0.5 mM	5.01 mL	25.06 mL	50.12 mL
1 mM	2.51 mL	12.53 mL	25.06 mL
5 mM	0.5 mL	2.51 mL	5.01 mL

*The above data is based on the productmolecular weight 399.05. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15828
M. Wt	399.05
Formula	C20H15Cl2N3O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1380087-86-4
Synonyms	CPI 268456, CPI268456
SMILES	C(N)(=O)C[C@@H]1N=C(C2=CC=C(Cl)C=C2)C2=CC(Cl)=CC=C2C2C(C)=NOC=21