CRT5
目录号: A22245
PKD 抑制剂
CRT5 (CRT0066051),一种吡嗪苯甲酰胺类化合物,是一种强效且选择性的PKD抑制剂,其IC50分别为PKD1的1 nM、PKD2的2 nM和PKD3的1.5 nM。
Discription | CRT5 (CRT0066051), a pyrazine benzamide, is a potent and selective PKD inhibitor with IC50 of 1 nM, 2 nM, and 1.5 nM for PKD1, PKD2, and PKD3, respectively. |
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目录号 | A22245 |
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分子式 | C28H30N4O2 |
分子量 | 454.57 |
CAS号 | 1034297-58-9 |
SMILES | O=C(NCCN(C)C)C1=CC=CC(C2=CC(C3=CC=C4C=C(OCC)C=CC4=C3)=C(N)N=C2)=C1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2