DPM-1001
目录号: A18674
PTP1B 抑制剂
DPM-1001 是一种强效的、特异性的、口服生物利用度高的非竞争性 蛋白酪氨酸磷酸酶(PTP1B)抑制剂,其 IC50 为 100 nM,是特异性 PTP1B 抑制剂 trodusquemine(MSI-1436;IC50=600 nM)的类似物。DPM-1001 具有抗糖尿病特性。
Discription | DPM-1001 is a potent, specific, orally bioavailable and non-competitive inhibitor of protein-tyrosine phosphatase (PTP1B) with an IC50 of 100 nM, an an analog of the specific PTP1B inhibitor trodusquemine (MSI-1436; IC50=600 nM). DPM-1001 has anti-diabetic property. |
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目录号 | A18674 |
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分子式 | C35H57N3O3 |
分子量 | 567.85 |
CAS号 | 1471172-27-6 |
SMILES | O[C@H]1[C@]2([H])[C@@](CC[C@@]3(C)[C@@]2([H])CC[C@]3([H])[C@H](C)CCC(OC)=O)([H])[C@]4(C)[C@@](C[C@H](NCCCCNCC5=CC=CC=N5)CC4)([H])C1 |
其他名称 | DPM-1001; DPM1001; DPM 1001 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2