DUBs-IN-3
目录号: A12830
USP7/USP8 抑制剂
DUBs-IN-3 是一种强效的去泛素化酶抑制剂,对 USP8 的 IC50 为 3.1 uM;对 USP7 的选择性超过 30 倍(IC50 > 100 uM)。
Discription | DUBs-IN-3 is a potent deubiquitinase enzyme inhibitor with IC50s of 3.1 uM for USP8; >30 fold selectivity over USP7 (IC50 > 100 uM). |
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目录号 | A12830 |
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分子式 | C16H9N5O |
分子量 | 287.28 |
CAS号 | 924296-17-3 |
SMILES | C=CCON=C1C2=CC=CC=C2C3=NC(=C(N=C31)C#N)C#N |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2