E-64
目录号: A13257
Cysteine Protease 抑制剂
E-64 是一种不可逆的、选择性的半胱氨酸蛋白酶抑制剂,对木瓜蛋白酶的 IC50 为 9 nM。
| Discription | E-64 is an irreversible and selective cysteine protease inhibitor with IC50 of 9 nM for papain. | ||
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| Targets |
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| 目录号 | A13257 |
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| 分子式 | C15H27N5O5 |
| 分子量 | 357.41 |
| CAS号 | 66701-25-5 |
| SMILES | CC(C)C[C@@H](C(=O)NCCCCN=C(N)N)NC(=O)[C@@H]1[C@H](O1)C(=O)O |
| 其他名称 | E64, E 64 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
| In vitro | DMSO | Warmed: 61 mg/mL (170.67 mM) | |
| Water | Warmed: 9 mg/mL (25.18 mM) | ||
| Ethanol | Insoluble | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 27.98 mL | 139.9 mL | 279.79 mL |
| 0.5 mM | 5.6 mL | 27.98 mL | 55.96 mL |
| 1 mM | 2.8 mL | 13.99 mL | 27.98 mL |
| 5 mM | 0.56 mL | 2.8 mL | 5.6 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2