EGFR-IN-5
目录号: A20082
EGFR 抑制剂
EGFR-IN-5 是一种 EGFR 抑制剂,其 IC50 分别针对 EGFR、EGFRL858R、EGFRL858R/T790M 和 EGFRL858R/T790M/C797S 为 10.4、1.1、34、7.2 nM。
Discription | EGFR-IN-5 is a EGFR inhibitor with IC50s of 10.4, 1.1, 34, 7.2 nM for EGFR, EGFRL858R, EGFRL858R/T790M, and EGFRL858R/T790M/C797S, respectively. | |||||
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Cell Research |
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目录号 | A20082 |
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分子式 | C31H38FN9O |
分子量 | 571.69 |
CAS号 | 2225887-26-1 |
SMILES | OCC(CC1)CCN1C2=NC(NC3=CC=C(F)C=C3)=NC(C=N4)=C2C=C4NC5=NC=C(N6CCC(N(C)C)CC6)C=C5 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2