Elacestrant
目录号: A12244
Estrogen receptor degrader
Elacestrant (RAD1901) 是一种口服可用的选择性雌激素受体降解剂(SERD),其对 ERα 和 ERβ 的 IC50 分别为 48 nM 和 870 nM。
Discription | Elacestrant (RAD1901) is an orally available selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively. | |||||
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Cell Research |
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目录号 | A12244 |
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分子式 | C30H38N2O2 |
分子量 | 458.63 |
CAS号 | 722533-56-4 |
SMILES | OC1=CC=C2C[C@H](C3=CC=C(OC)C=C3N(CC)CC4=CC=C(CCNCC)C=C4)CCC2=C1 |
其他名称 | RAD1901, RAD 1901, RAD-1901 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2