Eliprodil
目录号: A12946
NMDA 拮抗剂
Eliprodil 是一种非竞争性 NR2B-NMDA 受体拮抗剂(IC50=1 uM),对含 NR2A 和 NR2C 的受体的效力较低(IC50> 100 uM)。
Discription | Eliprodil is a non-competitive NR2B-NMDA receptor antagonist(IC50=1 uM), less potent for NR2A- and NR2C-containing receptors(IC50> 100 uM). |
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目录号 | A12946 |
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分子式 | C20H23ClFNO |
分子量 | 347.86 |
CAS号 | 119431-25-3 |
SMILES | ClC1=CC=C(C=C1)[C@H](CN2CCC(CC(C=C3)=CC=C3F)CC2)O |
其他名称 | SL-820715, SL820715, SL 820715 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 15 mg/mL (43.12 mM) | |
Water | Insoluble | ||
Ethanol | 5 mg/mL (14.37 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 28.75 mL | 143.74 mL | 287.47 mL |
0.5 mM | 5.75 mL | 28.75 mL | 57.49 mL |
1 mM | 2.87 mL | 14.37 mL | 28.75 mL |
5 mM | 0.57 mL | 2.87 mL | 5.75 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2